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HBI-3000

Structure via PubChem · Public domain (PubChem)

EntityQ5629032· pop 5· linked from 1 articles

Also known as sulcardine

HBI-3000 (sulcardine sulfate) is an experimental drug candidate that is currently in phase II of human clinical trials as an antiarrhythmic agent. Clinical investigation will test the safety and efficacy of HBI-3000 as a treatment for both atrial and ventricular arrhythmias.

Chemical data

Formula
C24H33N3O4S
Molecular weight
459.6 g/mol
IUPAC name
N-[[4-hydroxy-3,5-bis(pyrrolidin-1-ylmethyl)phenyl]methyl]-4-methoxybenzenesulfonamide
SMILES
COC1=CC=C(C=C1)S(=O)(=O)NCC2=CC(=C(C(=C2)CN3CCCC3)O)CN4CCCC4
InChIKey
SYZGIWXQGIBJGN-UHFFFAOYSA-N
XLogP
2.6
Polar surface area
90.5 Ų
H-bond donors
2
H-bond acceptors
7
Formal charge
0

via PubChem

Wikidata facts

Mass
459.219178
Show 2 more facts
chemical formula
C₂₄H₃₃N₃O₄S
canonical SMILES
COC1=CC=C(C=C1)S(=O)(=O)NCC2=CC(=C(C(=C2)CN3CCCC3)O)CN4CCCC4
Sources (2)

via Wikidata · CC0

~3 min read

Encyclopedic overview

8 sections
Contents
  • The molecular problem
  • Mechanism of action in ventricular myocytes
  • Studies
  • Animal model
  • Cellular isolation
  • Human studies
  • See also
  • References

{{Chembox | ImageFile = sulcardine.svg | ImageClass = skin-invert-image | ImageSize = 200px | PIN = N-({4-Hydroxy-3,5-bis[(pyrrolidin-1-yl)methyl]phenyl}methyl)-4-methoxybenzene-1-sulfonamide | OtherNames = |Section1= |Section2= |Section3= }}

HBI-3000 (sulcardine sulfate) is an experimental drug candidate that is currently in phase II of human clinical trials as an antiarrhythmic agent. Clinical investigation will test the safety and efficacy of HBI-3000 as a treatment for both atrial and ventricular arrhythmias.

Excerpted from Wikipedia’s “HBI-3000” article, available under the CC BY-SA 4.0 licence.

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