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demegestone

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EntityQ5255131· pop 9· linked from 397 articles

demegestone

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Also known as Lutionex

Demegestone, sold under the brand name Lutionex, is a progestin medication which was previously used to treat luteal insufficiency but is now no longer marketed. It is taken by mouth.

Chemical data

Formula
C21H28O2
Molecular weight
312.4 g/mol
IUPAC name
(8S,13S,14S,17S)-17-acetyl-13,17-dimethyl-1,2,6,7,8,11,12,14,15,16-decahydrocyclopenta[a]phenanthren-3-one
SMILES
CC(=O)[C@]1(CC[C@@H]2[C@@]1(CCC3=C4CCC(=O)C=C4CC[C@@H]23)C)C
InChIKey
JWAHBTQSSMYISL-MHTWAQMVSA-N
XLogP
2.8
Polar surface area
34.1 Ų
H-bond donors
0
H-bond acceptors
2
Formal charge
0

via PubChem

Drug data · ChEMBL

Max clinical phase
Phase 2
Molecule type
Small molecule

via ChEMBL · EBI

Wikidata facts

Mass
312.209
Show 4 more facts
chemical formula
C₂₁H₂₈O₂
isomeric SMILES
CC(=O)[C@]1(CC[C@@H]2[C@@]1(CCC3=C4CCC(=O)C=C4CC[C@@H]23)C)C
canonical SMILES
CC(=O)C1(CCC2C1(CCC3=C4CCC(=O)C=C4CCC23)C)C
Commons category
Demegestone
Sources (2)

via Wikidata · CC0

~4 min read

Encyclopedic overview

12 sections
Contents
  • Medical uses
  • Side effects
  • Pharmacology
  • Pharmacodynamics
  • Pharmacokinetics
  • Chemistry
  • History
  • Society and culture
  • Generic names
  • Brand names
  • Availability
  • References

Demegestone, sold under the brand name Lutionex, is a progestin medication which was previously used to treat luteal insufficiency but is now no longer marketed. It is taken by mouth.

Demegestone is a progestin, or a synthetic progestogen, and hence is an agonist of the progesterone receptor, the biological target of progestogens like progesterone. It has no androgenic activity.

Excerpted from Wikipedia’s “demegestone” article, available under the CC BY-SA 4.0 licence.

Available in 8 languages

via Wikidata sitelinks · CC0