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sulazepam

Structure via PubChem · Public domain (PubChem)

EntityQ7636056· pop 8· linked from 540 articles

Sulazepam is a benzodiazepine derivative. It is the thioamide derivative of diazepam. It is metabolised into diazepam, desmethyldiazepam and oxydiazepam. It has sedative, muscle relaxant, hypnotic, anticonvulsant and anxiolytic properties like those of other benzodiazepines. It was never marketed.

Chemical data

Formula
C16H13ClN2S
Molecular weight
300.8 g/mol
IUPAC name
7-chloro-1-methyl-5-phenyl-3H-1,4-benzodiazepine-2-thione
SMILES
CN1C(=S)CN=C(C2=C1C=CC(=C2)Cl)C3=CC=CC=C3
InChIKey
MWGWTOPCKLQYEU-UHFFFAOYSA-N
XLogP
3.6
Polar surface area
47.7 Ų
H-bond donors
0
H-bond acceptors
2
Formal charge
0

via PubChem

Drug data · ChEMBL

Max clinical phase
Phase 2
Molecule type
Small molecule

via ChEMBL · EBI

Wikidata facts

Mass
300.049
Show 3 more facts
chemical formula
C₁₆H₁₃ClN₂S
canonical SMILES
CN1C(=S)CN=C(C2=C1C=CC(=C2)Cl)C3=CC=CC=C3
Commons category
Sulazepam
Sources (2)

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~1 min read

Encyclopedic overview

3 sections
Contents
  • Synthesis
  • See also
  • References

Sulazepam is a benzodiazepine derivative. It is the thioamide derivative of diazepam. It is metabolised into diazepam, desmethyldiazepam and oxydiazepam. It has sedative, muscle relaxant, hypnotic, anticonvulsant and anxiolytic properties like those of other benzodiazepines. It was never marketed.

==Synthesis== thumb|center|400px|Sulazepam synthesis: Treatment of diazepam with phosphorus pentasulfide produces the corresponding thionamide, sulazepam. == See also == Uldazepam

Excerpted from Wikipedia’s “sulazepam” article, available under the CC BY-SA 4.0 licence.

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