Structure via PubChem · Public domain (PubChem)
meptazinol
Sign in to saveAlso known as Meptid
Meptazinol, sold under the brand name Meptid, is an opioid analgesic developed by Wyeth in the 1970s. Indications for use in moderate to severe pain, most commonly used to treat pain in obstetrics (childbirth).
Chemical data
- Formula
- C15H23NO
- Molecular weight
- 233.35 g/mol
- IUPAC name
- 3-(3-ethyl-1-methylazepan-3-yl)phenol
- SMILES
- CCC1(CCCCN(C1)C)C2=CC(=CC=C2)O
- InChIKey
- JLICHNCFTLFZJN-UHFFFAOYSA-N
- XLogP
- 3.4
- Polar surface area
- 23.5 Ų
- H-bond donors
- 1
- H-bond acceptors
- 2
- Formal charge
- 0
via PubChem
Drug data · ChEMBL
- Max clinical phase
- Approved
- Molecule type
- Small molecule
- Indications
- pain
via ChEMBL · EBI
Research
244 papers- Meptazinol.Lancet (London, England) · 1983
- Meptazinol.Lancet (London, England) · 1983
- Oral meptazinol--United Kingdom experience.Postgraduate medical journal · 1985
- Meptazinol. A review of its pharmacodynamic and pharmacokinetic properties and therapeutic efficacy.Drugs · 1985
- Asymmetric Total Synthesis of Meptazinol.The Journal of organic chemistry · 2022
via PubMed
Wikidata facts
- Subclass of
- chemical compound
- Mass
- 233.177964
- Has use
- medication
Show 4 more facts
- Commons category
- Meptazinol
- chemical formula
- C₁₅H₂₃NO
- canonical SMILES
- CCC1(CCCCN(C1)C)C2=CC(=CC=C2)O
- subject has role
- opioid antagonist
Sources (2)
via Wikidata · CC0
~1 min read
Encyclopedic overview
2 sectionsContents
- References
- External links
Meptazinol, sold under the brand name Meptid, is an opioid analgesic developed by Wyeth in the 1970s. Indications for use in moderate to severe pain, most commonly used to treat pain in obstetrics (childbirth).
Meptazinol is a 3-phenylazepane derivative, whereas the other phenazepanes like ethoheptazine and proheptazine are 4-phenylazepanes.
Excerpted from Wikipedia’s “meptazinol” article, available under the CC BY-SA 4.0 licence.