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Ricasetron
Sign in to saveRicasetron (BRL-46470) is a drug which acts as a selective antagonist at the serotonin 5-HT3 receptor. It has antiemetic effects as with other 5-HT3 antagonists, and also has anxiolytic effects significantly stronger than other related drugs, and with less side effects than benzodiazepine anxiolytics. However, it has never been developed for medical use.
Chemical data
Drug data · ChEMBL
- Max clinical phase
- Phase 2
- Molecule type
- Small molecule
via ChEMBL · EBI
Wikidata facts
- Subclass of
- chemical compound
- Mass
- 313.215412484
Show 3 more facts
- chemical formula
- C₁₉H₂₇N₃O
- canonical SMILES
- CC1(CN(c2c1cccc2)C(=O)N[CH]3C[CH]4CC[CH](C3)N4C)C
- isomeric SMILES
- CC1(CN(c2c1cccc2)C(=O)N[C@H]3C[C@H]4CC[C@@H](C3)N4C)C
Sources (2)
via Wikidata · CC0
~1 min read
Encyclopedic overview
2 sectionsContents
- See also
- References
Ricasetron (BRL-46470) is a drug which acts as a selective antagonist at the serotonin 5-HT3 receptor. It has antiemetic effects as with other 5-HT3 antagonists, and also has anxiolytic effects significantly stronger than other related drugs, and with less side effects than benzodiazepine anxiolytics. However, it has never been developed for medical use.
== See also == Zatosetron Bemesetron Tropanserin Tropisetron Granisetron
Excerpted from Wikipedia’s “Ricasetron” article, available under the CC BY-SA 4.0 licence.