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stampidine

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EntityQ7597499· pop 6· linked from 125 articles

stampidine

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Stampidine is an experimental nucleoside reverse transcriptase inhibitor (NRTI) with anti-HIV activity.

Chemical data

Formula
C20H23BrN3O8P
Molecular weight
544.3 g/mol
IUPAC name
methyl (2R)-2-[[(4-bromophenoxy)-[[(2S,5R)-5-(5-methyl-2,4-dioxopyrimidin-1-yl)-2,5-dihydrofuran-2-yl]methoxy]phosphoryl]amino]propanoate

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Wikidata facts

Mass
543.040613
Show 4 more facts
chemical formula
C₂₀H₂₃BrN₃O₈P
canonical SMILES
CC1=CN(C(=O)NC1=O)C2C=CC(O2)COP(=O)(NC(C)C(=O)OC)OC3=CC=C(C=C3)Br
isomeric SMILES
CC1=CN(C(=O)NC1=O)[C@H]2C=C[C@H](O2)COP(=O)(N[C@H](C)C(=O)OC)OC3=CC=C(C=C3)Br
Commons category
Stampidine
Sources (1)

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~4 min read

Article

2 sections
Contents
  • Preclinical pharmacology
  • References

{{Drugbox | verifiedrevid = 448073183 | IUPAC_name = methyl N-((4-bromophenoxy){[(2S,5R)-5-(5-methyl-2,4-dioxo-3,4-dihydropyrimidin-1(2H)-yl)-2,5-dihydrofuran-2-yl]methoxy}phosphoryl)-D-alaninate | image = Stampidine structure.svg | image_class = skin-invert-image | alt = Skeletal formula of stampidine | width = 250 | image2 = Stampidine-3D-balls.png | image_class2 = bg-transparent | alt2 = Ball-and-stick model of the stampidine molecule

| tradename = | pregnancy_AU = | pregnancy_US = | pregnancy_category = | legal_AU = | legal_CA = | legal_UK = | legal_US = | legal_status = | routes_of_administration =

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