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dazopride
Sign in to saveDazopride (AHR-5531) is an antiemetic and gastroprokinetic agent of the benzamide class which was never marketed. It acts as a 5-HT3 receptor antagonist and 5-HT4 receptor agonist. In addition to its gastrointestinal effects, dazopride facilitates learning and memory in mice.
Chemical data
- Formula
- C15H23ClN4O2
- Molecular weight
- 326.82 g/mol
- IUPAC name
- 4-amino-5-chloro-N-(1,2-diethylpyrazolidin-4-yl)-2-methoxybenzamide
- SMILES
- CCN1CC(CN1CC)NC(=O)C2=CC(=C(C=C2OC)N)Cl
- InChIKey
- YFXIKEZOBJFVAQ-UHFFFAOYSA-N
- XLogP
- 2
- Polar surface area
- 70.8 Ų
- H-bond donors
- 2
- H-bond acceptors
- 5
- Formal charge
- 0
via PubChem
Drug data · ChEMBL
- Max clinical phase
- Phase 2
- Molecule type
- Small molecule
via ChEMBL · EBI
Wikidata facts
- Subclass of
- chemical compound
- Mass
- 326.151
Show 3 more facts
- canonical SMILES
- CCN1CC(CN1CC)NC(=O)C2=CC(=C(C=C2OC)N)Cl
- chemical formula
- C₁₅H₂₃ClN₄O₂
- Commons category
- Dazopride
Sources (2)
via Wikidata · CC0
~1 min read
Encyclopedic overview
2 sectionsContents
- See also
- References
Dazopride (AHR-5531) is an antiemetic and gastroprokinetic agent of the benzamide class which was never marketed. It acts as a 5-HT3 receptor antagonist and 5-HT4 receptor agonist. In addition to its gastrointestinal effects, dazopride facilitates learning and memory in mice.
== See also == Antiemetic Benzamide
Excerpted from Wikipedia’s “dazopride” article, available under the CC BY-SA 4.0 licence.
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