E-55888
Sign in to saveAlso known as N,N-Dimethyl-2-[3-(1,3,5-trimethylpyrazol-4-yl)phenyl]ethanamine, E55888, E 55888
E-55888 is a drug developed by Esteve, which acts as a potent and selective full agonist at the 5HT7 serotonin receptor, and is used for investigating the role of 5-HT7 receptors in the perception of pain. When administered by itself, E-55888 is anti-hyperalgesic but not analgesic, but when administered alongside morphine, E-55888 was found to significantly increase the analgesic effects.
Wikidata facts
- Subclass of
- chemical compound
- Mass
- 257.189198
Show 2 more facts
- chemical formula
- C₁₆H₂₃N₃
- canonical SMILES
- CC1=C(C(=NN1C)C)C2=CC(=CC=C2)CCN(C)C
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Encyclopedic overview
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- See also
- References
E-55888 is a drug developed by Esteve, which acts as a potent and selective full agonist at the 5HT7 serotonin receptor, and is used for investigating the role of 5-HT7 receptors in the perception of pain. When administered by itself, E-55888 is anti-hyperalgesic but not analgesic, but when administered alongside morphine, E-55888 was found to significantly increase the analgesic effects.
==See also== AS-19 LP-12 LP-44 LP-211
Excerpted from Wikipedia’s “E-55888” article, available under the CC BY-SA 4.0 licence.