Structure via PubChem · Public domain (PubChem)
enpiprazole
Sign in to saveEnpiprazole (INN, BAN) is an anxiolytic drug of the phenylpiperazine group that was never marketed. It produces anxiolytic-like effects in animals, though these effects appear to be biphasic and may reverse at high doses. It is known to produce ortho-chlorophenylpiperazine (oCPP) as a metabolite.
Chemical data
- Formula
- C16H21ClN4
- Molecular weight
- 304.82 g/mol
- IUPAC name
- 1-(2-chlorophenyl)-4-[2-(1-methylpyrazol-4-yl)ethyl]piperazine
- SMILES
- CN1C=C(C=N1)CCN2CCN(CC2)C3=CC=CC=C3Cl
- InChIKey
- WBFVWQJVMMIQFI-UHFFFAOYSA-N
- XLogP
- 2.8
- Polar surface area
- 24.3 Ų
- H-bond donors
- 0
- H-bond acceptors
- 3
- Formal charge
- 0
via PubChem
Drug data · ChEMBL
- Max clinical phase
- Phase 2
- Molecule type
- Small molecule
via ChEMBL · EBI
Wikidata facts
- Subclass of
- chemical compound
- Mass
- 304.145
Show 2 more facts
- chemical formula
- C₁₆H₂₁ClN₄
- canonical SMILES
- CN1C=C(C=N1)CCN2CCN(CC2)C3=CC=CC=C3Cl
Sources (2)
via Wikidata · CC0
~1 min read
Encyclopedic overview
2 sectionsContents
- See also
- References
Enpiprazole (INN, BAN) is an anxiolytic drug of the phenylpiperazine group that was never marketed. It produces anxiolytic-like effects in animals, though these effects appear to be biphasic and may reverse at high doses. It is known to produce ortho-chlorophenylpiperazine (oCPP) as a metabolite.
==See also== Acaprazine Enciprazine Lorpiprazole Mepiprazole Tolpiprazole
Excerpted from Wikipedia’s “enpiprazole” article, available under the CC BY-SA 4.0 licence.