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lufuradom

Structure via PubChem · Public domain (PubChem)

EntityQ6699691· pop 9· linked from 871 articles

Lufuradom (INN) is a drug and benzodiazepine derivative which, unlike other benzodiazepines, is described as an analgesic. Similarly to its analogue tifluadom, it was never marketed.

Chemical data

Formula
C22H20FN3O2
Molecular weight
377.4 g/mol
IUPAC name
N-[(8-fluoro-1-methyl-5-phenyl-2,3-dihydro-1,4-benzodiazepin-2-yl)methyl]furan-3-carboxamide
SMILES
CN1C(CN=C(C2=C1C=C(C=C2)F)C3=CC=CC=C3)CNC(=O)C4=COC=C4
InChIKey
QJSCDZOUCFWCKD-UHFFFAOYSA-N
XLogP
3
Polar surface area
57.8 Ų
H-bond donors
1
H-bond acceptors
5
Formal charge
0

via PubChem

Drug data · ChEMBL

Max clinical phase
Phase 2
Molecule type
Small molecule

via ChEMBL · EBI

Wikidata facts

Mass
377.154
Show 3 more facts
chemical formula
C₂₂H₂₀FN₃O₂
canonical SMILES
CN1C(CN=C(C2=C1C=C(C=C2)F)C3=CC=CC=C3)CNC(=O)C4=COC=C4
Commons category
Lufuradom
Sources (1)

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Encyclopedic overview

2 sections
Contents
  • See also
  • References

Lufuradom (INN) is a drug and benzodiazepine derivative which, unlike other benzodiazepines, is described as an analgesic. Similarly to its analogue tifluadom, it was never marketed.

== See also == Tifluadom GYKI-52895, structural benzodiazepine which is a dopamine reuptake inhibitor without GABAergic function GYKI-52,466, structural benzodiazepine which is an AMPAkine and glutamate antagonist without GABAergic function

Excerpted from Wikipedia’s “lufuradom” article, available under the CC BY-SA 4.0 licence.

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