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پلریکسافور

Structure via PubChem · Public domain (PubChem)

EntityQ905835· pop 12· linked from 147 articles

پلریکسافور

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Also known as AMD 3100, AMD3100, bicyclam JM-2987, JM 3100, Mozobil®

ترکیب شیمیایی

Chemical data

Formula
C28H54N8
Molecular weight
502.8 g/mol
IUPAC name
1-[[4-(1,4,8,11-tetrazacyclotetradec-1-ylmethyl)phenyl]methyl]-1,4,8,11-tetrazacyclotetradecane
SMILES
C1CNCCNCCCN(CCNC1)CC2=CC=C(C=C2)CN3CCCNCCNCCCNCC3
InChIKey
YIQPUIGJQJDJOS-UHFFFAOYSA-N
XLogP
0
Polar surface area
78.7 Ų
H-bond donors
6
H-bond acceptors
8
Formal charge
0

via PubChem

Drug data · ChEMBL

Max clinical phase
Approved
Molecule type
Small molecule
First approval
2008
Admin. routes
parenteral
Indications
acute graft vs. host disease, multiple myeloma, acute myeloid leukemia, lymphoma

via ChEMBL · EBI

Wikidata facts

Mass
502.447
Has use
medication
Show 6 more facts
chemical formula
C₂₈H₅₄N₈
canonical SMILES
C1CNCCNCCCN(CCNC1)CC2=CC=C(C=C2)CN3CCCNCCNCCCNCC3
defined daily dose
16.8
medical condition treated
multiple myeloma
physically interacts with
C-X-C motif chemokine receptor 4
Commons category
Plerixafor
Sources (7)

via Wikidata · CC0