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gestodene
EntityQ408289· pop 12· linked from 1,019 articles

Also known as SH B 331, SID144205785, SH b 331

Gestodene, sold under the brand names Femodene and Minulet among others, is a progestin medication which is used in birth control pills for women. It is also used in menopausal hormone therapy. The medication is available almost exclusively in combination with an estrogen. It is taken by mouth.

Wikidata facts

Mass
310.193
Show 6 more facts
chemical formula
C₂₁H₂₆O₂
World Health Organisation international non-proprietary name
gestodene
isomeric SMILES
CC[C@]12CC[C@H]3[C@H]([C@@H]1C=C[C@]2(C#C)O)CCC4=CC(=O)CC[C@H]34
canonical SMILES
CCC12CCC3C(C1C=CC2(C#C)O)CCC4=CC(=O)CCC34
MCN code
2937.23.92
Commons category
Gestodene
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~11 min read

Article

23 sections
Contents
  • Medical uses
  • Available forms
  • Contraindications
  • Side effects
  • Overdose
  • Contraindications
  • Pharmacology
  • Pharmacodynamics
  • Progestogenic activity
  • Androgenic activity
  • Glucocorticoid activity
  • Antimineralocorticoid activity
  • Other activities
  • Pharmacokinetics
  • Chemistry
  • Synthesis
  • History
  • Society and culture
  • Generic names
  • Brand names
  • Availability
  • References
  • Further reading

Gestodene, sold under the brand names Femodene and Minulet among others, is a progestin medication which is used in birth control pills for women. It is also used in menopausal hormone therapy. The medication is available almost exclusively in combination with an estrogen. It is taken by mouth.

Side effects of the combination of an estrogen and gestodene include menstrual irregularities, headaches, nausea, breast tenderness, mood changes, and others. Gestodene is a progestin, or a synthetic progestogen, and hence is an agonist of the progesterone receptor, the biological target of progestogens like progesterone. It has weak androgenic activity, weak antimineralocorticoid activity, and weak glucocorticoid activity.

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