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nicodicodine

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Nicodicodine is an opioid developed as a cough suppressant and analgesic. Synthesized in 1904, it is not commonly used, but has activity similar to other opioids. Nicodicodine is metabolised in the liver by demethylation to produce 6-nicotinoyldihydromorphine, and subsequently further metabolised to dihydromorphine. Since the final active metabolite is the slightly stronger opiate dihydromorphine rather than morphine, nicodicodine can be expected to be marginally more potent and longer acting than nicocodeine. Side effects are similar to those of other opioids and include itching, nausea and r

Key facts

Drug.Watchedfields
changed
Drug.Verifiedfields
changed
Drug.verifiedrevid
447732381
Drug.IUPAC_name
(5alpha,6alpha)-3-Methoxy-17-methyl-4,5-epoxymorphinan-6-yl pyridine-3-carboxylate
Drug.image
Nicodicodeine.svg
Drug.image_class
skin-invert-image
Drug.alt
Structural formula
Drug.width
210
Drug.image2
Nicodicodeine molecule ball.png
Drug.image_class2
bg-transparent
Drug.alt2
Ball-and-stick model
Drug.width2
220
Drug.legal_AU
S2
Drug.legal_BR
A2
Drug.legal_DE
Anlage II
Drug.legal_UK
Class B
Drug.legal_UN
narcotic schedules i and iii
Drug.routes_of_administration
Oral, intravenous

via Wikipedia infobox

Wikidata facts

Mass
406.189
Show 4 more facts
chemical formula
C₂₄H₂₆N₂O₄
canonical SMILES
CN1CCC23C4C1CC5=C2C(=C(C=C5)OC)OC3C(CC4)OC(=O)C6=CN=CC=C6
isomeric SMILES
CN1CC[C@]23[C@@H]4[C@H]1CC5=C2C(=C(C=C5)OC)O[C@H]3[C@H](CC4)OC(=O)C6=CN=CC=C6
Commons category
Nicodicodeine
Sources (2)

via Wikidata · CC0

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Encyclopedic overview

1 sections
Contents
  • References

Nicodicodine is an opioid developed as a cough suppressant and analgesic. Synthesized in 1904, it is not commonly used, but has activity similar to other opioids. Nicodicodine is metabolised in the liver by demethylation to produce 6-nicotinoyldihydromorphine, and subsequently further metabolised to dihydromorphine. Since the final active metabolite is the slightly stronger opiate dihydromorphine rather than morphine, nicodicodine can be expected to be marginally more potent and longer acting than nicocodeine. Side effects are similar to those of other opioids and include itching, nausea and respiratory depression.

==References==

Excerpted from Wikipedia’s “nicodicodine” article, available under the CC BY-SA 4.0 licence.