phaclofen
Sign in to savePhaclofen, or phosphonobaclofen, is a selective antagonist for the GABAB receptor. It was the first selective GABAB antagonist discovered, but its utility was limited by the fact that it does not cross the blood brain barrier.
Wikidata facts
- Mass
- 249.032158
Show 2 more facts
- chemical formula
- C₉H₁₃ClNO₃P
- canonical SMILES
- C1=CC(=CC=C1C(CN)CP(=O)(O)O)Cl
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Phaclofen, or phosphonobaclofen, is a selective antagonist for the GABAB receptor. It was the first selective GABAB antagonist discovered, but its utility was limited by the fact that it does not cross the blood brain barrier.
==References==
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