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ertapenem

Structure via PubChem · Public domain (PubChem)

EntityQ553220· pop 24· linked from 242 articles

Also known as (4R,5S,6S)-3-((3S,5S)-5-((3-Carboxyphenyl)carbamoyl)pyrrolidin-3-ylthio)-6-((R)-1-hydroxyethyl)-4-methyl-7-oxo-1-aza-bicyclo[3.2.0]hept-2-ene-2-carboxylic acid, (1R,5S,6S,8R,2'S,4's)-2-(2-(3-carboxyphenylcarbamoyl)pyrrolidin-4-ylthio)-6-(1-hydroxyethyl)-1-methylcarbapenem-3-carboxylic acid

Ertapenem, sold under the brand name Invanz, is a carbapenem antibiotic medication used for the treatment of infections of the abdomen, the lungs, the upper part of the female reproductive system, and the diabetic foot.

Key facts

Drug.H
25
Drug.N
3
Drug.O
7
Drug.S
1
Drug.Verifiedfields
changed
Drug.verifiedrevid
461095141
Drug.image
Ertapenem skeletal structure.svg
Drug.image_class
skin-invert-image
Drug.image2
Ertapenem ball-and-stick model.png
Drug.image_class2
bg-transparent
Drug.tradename
Invanz
Drug.MedlinePlus
a614001
Drug.DailyMedID
Ertapenem
Drug.pregnancy_AU
B3
Drug.routes_of_administration
Intramuscular, intravenous
Drug.ATC_prefix
J01
Drug.ATC_suffix
DH03
Drug.legal_AU
S4

via Wikipedia infobox

Chemical data

Formula
C22H25N3O7S
Molecular weight
475.5 g/mol
IUPAC name
(4R,5S,6S)-3-[(3S,5S)-5-[(3-carboxyphenyl)carbamoyl]pyrrolidin-3-yl]sulfanyl-6-[(1R)-1-hydroxyethyl]-4-methyl-7-oxo-1-azabicyclo[3.2.0]hept-2-ene-2-carboxylic acid
SMILES
C[C@@H]1[C@@H]2[C@H](C(=O)N2C(=C1S[C@H]3C[C@H](NC3)C(=O)NC4=CC=CC(=C4)C(=O)O)C(=O)O)[C@@H](C)O
InChIKey
JUZNIMUFDBIJCM-ANEDZVCMSA-N
XLogP
-1.5
Polar surface area
182 Ų
H-bond donors
5
H-bond acceptors
9
Formal charge
0

via PubChem

Research

2,591 papers

via PubMed

Wikidata facts

Mass
475.141321
Manufacturer
Pfizer
Has use
medication
Show 9 more facts
medical condition treated
pyelonephritis
chemical formula
C₂₂H₂₅N₃O₇S
isomeric SMILES
C[C@@H]1[C@@H]2[C@H](C(=O)N2C(=C1S[C@H]3C[C@H](NC3)C(=O)NC4=CC=CC(=C4)C(=O)O)C(=O)O)[C@@H](C)O
canonical SMILES
CC1C2C(C(=O)N2C(=C1SC3CC(NC3)C(=O)NC4=CC=CC(=C4)C(=O)O)C(=O)O)C(C)O
World Health Organisation international non-proprietary name
ertapenem
defined daily dose
1
subject has role
bactericide
stylized name
INVanz
Commons category
Ertapenem
Sources (7)

via Wikidata · CC0

~8 min read

Encyclopedic overview

13 sections
Contents
  • Medical uses
  • Contraindications
  • Side effects
  • Overdose
  • Interactions
  • Pharmacology
  • Mechanism of action
  • Susceptible bacteria
  • Resistance
  • Pharmacokinetics
  • Comparison with other antibiotics
  • History
  • References

Ertapenem, sold under the brand name Invanz, is a carbapenem antibiotic medication used for the treatment of infections of the abdomen, the lungs, the upper part of the female reproductive system, and the diabetic foot.

The most common side effects include diarrhoea, nausea, headache, and problems around the area where the medicine is infused. It can significantly reduce the concentrations of valproic acid, an anti-seizure medication, in the blood to the point where it loses its effectiveness.

Excerpted from Wikipedia’s “ertapenem” article, available under the CC BY-SA 4.0 licence.

Gallery (5)