Skip to content
EntityQ416331· pop 24· linked from 394 articles

pentoxifylline

Sign in to save

Also known as BL-191, Trental®, Pentoxifyllin, Pentoxifyllinum, Oxpentifylline, Pentoxifilina

Pentoxifylline, also known as oxpentifylline, is a xanthine derivative used as a drug to treat muscle pain in people with peripheral artery disease. It was approved for medical use in 1984 and is available as generic and sold under many brand names worldwide like Trental.

Key facts

Drug.pregnancy_AU
B1
Drug.Watchedfields
changed
Drug.verifiedrevid
464198476
Drug.IUPAC_name
3,7-Dimethyl-1-(5-oxohexyl)purine-2,6-dione
Drug.image
Pentoxifylline.svg
Drug.image_class
skin-invert-image
Drug.width
180
Drug.image2
Pentoxifylline xtal 2005 ball-and-stick.png
Drug.image_class2
bg-transparent
Drug.width2
200
Drug.tradename
Trental, many other names worldwide
Drug.MedlinePlus
a685027
Drug.licence_US
Pentoxifylline
Drug.pregnancy_US
C
Drug.legal_AU
S4
Drug.legal_CA
Rx-only
Drug.legal_UK
POM
Drug.legal_US
Rx-only

via Wikipedia infobox

Research

6,081 papers

via PubMed

Wikidata facts

Mass
278.138
Show 5 more facts
chemical formula
C₁₃H₁₈N₄O₃
Commons category
Pentoxifylline
canonical SMILES
CC(=O)CCCCN1C(=O)C2=C(N=CN2C)N(C1=O)C
half-life
0.6
stylized name
TRENtal
Sources (6)

via Wikidata · CC0

~7 min read

Article

7 sections
Contents
  • Medical uses
  • Adverse effects
  • Mechanism
  • Research
  • See also
  • References
  • External links

Pentoxifylline, also known as oxpentifylline, is a xanthine derivative used as a drug to treat muscle pain in people with peripheral artery disease. It was approved for medical use in 1984 and is available as generic and sold under many brand names worldwide like Trental.

== Medical uses == Its primary use in medicine is to reduce pain, cramping, numbness, or weakness in the arms or legs which occurs due to intermittent claudication, a form of muscle pain resulting from peripheral artery diseases. This is its only FDA, MHRA and TGA-labelled indication. However, pentoxifylline is also recommended for off-label use as an adjunct to compression bandaging for the treatment of chronic venous leg ulcers by the Scottish Intercollegiate Guidelines Network (SIGN) as this has been shown to improve healing rates.

Connections

Categories