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Sunepitron
Sign in to saveSunepitron (developmental code name CP-93,393) is a combined 5-HT1A receptor agonist and α2-adrenergic receptor antagonist. It was previously under development by Pfizer for the treatment of depression and anxiety. It made it to phase III clinical trials before being discontinued.
In the Vinony graph
Vinony's link graph records 1,704 inbound references to Sunepitron, and connects out to propranolol, N-methylserotonin and atenolol.
It is catalogued under topics including 5-HT1A agonists, Abandoned drugs and Alpha-2 blockers.
Vinony links it to 5 Wikipedia language editions.
Chemical data
- Formula
- C17H23N5O2
- Molecular weight
- 329.4 g/mol
- IUPAC name
- 1-[(2-pyrimidin-2-yl-1,3,4,6,7,8,9,9a-octahydropyrido[1,2-a]pyrazin-7-yl)methyl]pyrrolidine-2,5-dione
- SMILES
- C1CC2CN(CCN2CC1CN3C(=O)CCC3=O)C4=NC=CC=N4
- InChIKey
- UXWBIYCPUVWKHP-UHFFFAOYSA-N
- XLogP
- 0.2
- Polar surface area
- 69.6 Ų
- H-bond donors
- 0
- H-bond acceptors
- 6
- Formal charge
- 0
via PubChem
Wikidata facts
- Subclass of
- chemical compound
- Mass
- 329.185175
Show 2 more facts
- chemical formula
- C₁₇H₂₃N₅O₂
- canonical SMILES
- C1CC2CN(CCN2CC1CN3C(=O)CCC3=O)C4=NC=CC=N4
Sources (1)
via Wikidata · CC0
~2 min read
Encyclopedic overview
4 sectionsContents
- Chemistry
- Synthesis
- See also
- References
{{Drugbox | IUPAC_name = 1-{[2-(pyrimidin-2-yl)octahydro-2H-pyrido[1,2-a]pyrazin-7-yl]methyl}pyrrolidine-2,5-dione | image = Sunepitron.png | image_class = skin-invert-image | width =
| tradename = | pregnancy_category = | legal_status = | routes_of_administration = Oral
Excerpted from Wikipedia’s “Sunepitron” article, available under the CC BY-SA 4.0 licence.